Cannabis Ruderalis

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* [[5F-CUMYL-PINACA]]
* [[5F-CUMYL-PINACA]]
* [[5F-SDB-006]]
* [[5F-SDB-006]]
* [[CUMYL-PINACA]]
* [[CUMYL-THPINACA]]
* [[CUMYL-THPINACA]]
* [[SDB-006]]
* [[SDB-006]]

Revision as of 10:24, 11 July 2015

CUMYL-PICA
Identifiers
  • 1-pentyl-N-(2-phenylpropan-2-yl)-1H-indole-3-carboxamide
CAS Number
Chemical and physical data
FormulaC23H28N2O
Molar mass348.49 g/mol g·mol−1
3D model (JSmol)
  • O=C(NC(C)(C)C1=CC=CC=C1)C2=CN(CCCCC)C3=C2C=CC=C3
  • InChI=1S/C23H28N2O/c1-4-5-11-16-25-17-20(19-14-9-10-15-21(19)25)22(26)24-23(2,3)18-12-7-6-8-13-18/h6-10,12-15,17H,4-5,11,16H2,1-3H3,(H,24,26)
  • Key:RCXFMWJQOYCIQU-UHFFFAOYSA-N

CUMYL-PICA (SGT-56) is an indole-3-carboxamide based synthetic cannabinoid. It is the α,α-dimethylbenzyl analogue of SDB-006.[1] It was briefly sold in New Zealand during 2013 as an ingredient of at the time legal synthetic cannabis products, but the product containing CUMYL-BICA and CUMYL-PICA was denied an interim licensing approval under the Psychoactive Substances regulatory scheme, due to reports of adverse events in consumers.[2] CUMYL-PICA acts as a potent agonist for the cannabinoid receptors, with approximately 20x selectivity for CB1, having an EC50 of 0.66nM for human CB1 receptors and 13nM for human CB2 receptors.[3]

See also

References

  1. ^ "CUMYL-PICA". Cayman Chemical. Retrieved 8 July 2015.
  2. ^ The Risk Assessment Score Table. New Zealand Ministry of Health, 27 September 2013
  3. ^ Bowden; et al. (11 April 2013). "Patent WO 2014167530 - Cannabinoid compounds". New Zealand Patent application 623626. Retrieved 11 July 2015. {{cite web}}: Explicit use of et al. in: |author= (help)

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